Total regioselective control of tartaric acid

Jan Spengler; Ana I. Fernández-Llamazares; Javier Ruiz-Rodríguez; Klaus Burger; Fernando Albericio

doi:10.1021/jo101001s

Total regioselective control of tartaric acid

Jan Spengler
, Ana I. Fernández-Llamazares
, Javier Ruiz-Rodríguez
, Klaus Burger
, Fernando Albericio

Research output: Contribution to journal › Article › peer-review

5 Scopus citations

Abstract

An efficient strategy to synthesize tartaric acid building blocks for totally regioselective transformations or derivatizations was disclosed. Starting from l-tartaric acid or l-dimethyl tartrate, respectively, we obtained type I and II building blocks with orthogonal sets of protecing groups (4-8 steps, 38-56% overall yield).

Original language	English
Pages (from-to)	5746-5749
Number of pages	4
Journal	Journal of Organic Chemistry
Volume	75
Issue number	16
DOIs	https://doi.org/10.1021/jo101001s
State	Published - 20 Aug 2010
Externally published	Yes

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10.1021/jo101001s

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title = "Total regioselective control of tartaric acid",

abstract = "An efficient strategy to synthesize tartaric acid building blocks for totally regioselective transformations or derivatizations was disclosed. Starting from l-tartaric acid or l-dimethyl tartrate, respectively, we obtained type I and II building blocks with orthogonal sets of protecing groups (4-8 steps, 38-56\% overall yield).",

author = "Jan Spengler and Fern{\'a}ndez-Llamazares, \{Ana I.\} and Javier Ruiz-Rodr{\'i}guez and Klaus Burger and Fernando Albericio",

year = "2010",

month = aug,

day = "20",

doi = "10.1021/jo101001s",

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pages = "5746--5749",

journal = "Journal of Organic Chemistry",

issn = "0022-3263",

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TY - JOUR

T1 - Total regioselective control of tartaric acid

AU - Spengler, Jan

AU - Fernández-Llamazares, Ana I.

AU - Ruiz-Rodríguez, Javier

AU - Burger, Klaus

AU - Albericio, Fernando

PY - 2010/8/20

Y1 - 2010/8/20

N2 - An efficient strategy to synthesize tartaric acid building blocks for totally regioselective transformations or derivatizations was disclosed. Starting from l-tartaric acid or l-dimethyl tartrate, respectively, we obtained type I and II building blocks with orthogonal sets of protecing groups (4-8 steps, 38-56% overall yield).

AB - An efficient strategy to synthesize tartaric acid building blocks for totally regioselective transformations or derivatizations was disclosed. Starting from l-tartaric acid or l-dimethyl tartrate, respectively, we obtained type I and II building blocks with orthogonal sets of protecing groups (4-8 steps, 38-56% overall yield).

UR - https://www.scopus.com/pages/publications/77955678953

U2 - 10.1021/jo101001s

DO - 10.1021/jo101001s

M3 - Artículo

C2 - 20704449

AN - SCOPUS:77955678953

SN - 0022-3263

VL - 75

SP - 5746

EP - 5749

JO - Journal of Organic Chemistry

JF - Journal of Organic Chemistry

IS - 16

ER -

Total regioselective control of tartaric acid

Abstract

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